Aromasin 12.5mg/30tabs - Exemestane - Innovagen

• Classification: Aromatase Inhibitor
• Hepatotoxicity None
• Active Half-life: 9 hours
• Recommended Dosage: 6.25-25 mg/day

Aromatase Inhibitors General Info

Aromatase Inhibitors are drugs that block the enzyme aromatase. The aromatase enzyme converts androgens into estrogen.

Examples of Estrogenic activity levels of popular compounds.

Testosterone - Aromatized by the body -Moderate estrogenic activity

Dianabol - Aromatized by the body - Moderate estrogenic activity

Boldenone - Aromatized by the body - Low estrogenic activity

Nandrolone - (Low) Aromatized by the body - Low estrogenic activity

Masterone - Not Aromatized by the body - No estrogenic activity

Winstrol - Not Aromatized by the body - No estrogenic activity

Anavar - Not Aromatized by the body - No estrogenic activity

Anadrol - Not Aromatized by the body - High estrogenic activity

Aromasin General Info

Aromatase Inhibitor Aromasin is an irreversible steroidal inhibitor that forms a deactivating bond with the aromatase enzyme. Aromasin is FDA approved drug, and it is widely used in breast cancer treatment of postmenopausal women and gynecomastia in men.

Aromasin in Sports

Male athletes and bodybuilders use Aromasin to prevent estrogenic side effects such as gynecomastia, water retention, fat build-up. Another important benefit of Aromasin is that it lowers the Sex Hormone Binding Globulin (SHBG) by more than 20%.SHBG binds to testosterone and reduces the free testosterone levels.

Please note 

Some compounds do not convert to estrogen however have a high level of estrogenic activity. An excellent example of such compound is Oxymetholone. Anti-aromatase compounds Arimidex, Femara, or Aromasin, will not be effective. To avoid the estrogenic side effects, we recommend using anti-estrogens such as Nolvadex and Clomid.

Administration Men

Recommended dosage range 6.25-25 mg/day

Aromasin Pharmacokinetics

Administration of 25 mg dose of Aromasin.

• 24 hours estrogen levels reduced by 70-80%
• 72 hours after the administration -estrogen levels are 40% lower than the baseline
• 120 hours after administration-estrogen levels returned to baseline levels

As you can see, Aromasin is a very potent compound, and dosages are user unique. Proper dosages are only decided by blood work. The best practice is to take Aromasin at 6.25 mg x2 times a day for 7-10 days and, after that, get blood work done. Once you know your estrogen levels, you can higher or lower the Aromasin dosage. Please plan your Aromasin dosage carefully, get your blood work done, and, if possible, seek professional advice.